Document quand l'auteur est "Lubell, William D"

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Wei, Xiaozheng; Diarra, Sitan; Douchez, Antoine; Dallagnol, Juliana C; Hébert, Terence E; Chatenet, David ORCID: https://orcid.org/0000-0002-7270-4328 et Lubell, William D (2023). Urotensin II Receptor Modulation with 1,3,4-Benzotriazepin-2-one Tetrapeptide Mimics Journal of Medicinal Chemistry , vol. 66 , nº 20. pp. 14241-14262. DOI: 10.1021/acs.jmedchem.3c01307.

Merlino, Francesco; Billard, Étienne; Yousif, Ali Munaim; Di Maro, Salvatore; Brancaccio, Diego; Abate, Luigi; Carotenuto, Alfonso; Bellavita, Rosa; d'Emmanuele di Villa Bianca, Roberta; Santicioli, Paola; Marinelli, Luciana; Novellino, Ettore; Hébert, Terence E; Lubell, William D; Chatenet, David et Grieco, Paolo (2019). Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides Journal of Medicinal Chemistry , vol. 62 , nº 3. pp. 1455-1467. DOI: 10.1021/acs.jmedchem.8b01601.

Strack, Martin; Billard, Étienne; Chatenet, David et Lubell, William D (2017). Urotensin core mimics that modulate the biological activity of urotensin-II related peptide but not urotensin-II Bioorganic and Medicinal Chemistry Letters , vol. 27 , nº 15. pp. 3412-3416. DOI: 10.1016/j.bmcl.2017.05.088.

Douchez, Antoine; Billard, Étienne; Hébert, Terence E; Chatenet, David et Lubell, William D (2017). Design, Synthesis, and Biological Assessment of Biased Allosteric Modulation of the Urotensin II Receptor Using Achiral 1,3,4-Benzotriazepin-2-one Turn Mimics Journal of Medicinal Chemistry , vol. 60 , nº 23. pp. 9838-9859. DOI: 10.1021/acs.jmedchem.7b01525.

Merlino, Francesco; Yousif, Ali Munaim; Billard, Étienne; Dufour-Gallant, Julien; Turcotte, Stéphane; Grieco, Paolo; Chatenet, David et Lubell, William D (2016). Urotensin II(4-11) Azasulfuryl Peptides: Synthesis and Biological Activity Journal of Medicinal Chemistry , vol. 59 , nº 10. pp. 4740-4752. DOI: 10.1021/acs.jmedchem.6b00108.

Dufour-Gallant, Julien; Chatenet, David et Lubell, William D (2015). De Novo Conception of Small Molecule Modulators Based on Endogenous Peptide Ligands: Pyrrolodiazepin-2-one gamma-Turn Mimics That Differentially Modulate Urotensin II Receptor-Mediated Vasoconstriction ex Vivo Journal of Medicinal Chemistry , vol. 58 , nº 11. pp. 4624-37. DOI: 10.1021/acs.jmedchem.5b00162.

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Lubell, William D; Wei, Xiaozheng; Diarra, Sitan; Douchez, Antoine; Dallagnol, Juliana C; Harvey-Lavoie, Simonne; Hébert, Terence E et Chatenet, David ORCID: https://orcid.org/0000-0002-7270-4328 (2024). Tetrasubstituted benzotriazepinones act as β-turn mimics without stereogenic carbons exhibiting allosteric modulation of the urotensin II receptor In: 37th European Peptide Symposium 14th International Peptide Symposium, August 25-29, 2024, Florence, Italy.