Document quand l'auteur est "Billard, Étienne"

Nassour, Hassan; Pétrin, Darlaine; Devost, Dominic; Billard, Étienne; Sleno, Rory; Hébert, Terence E et Chatenet, David ORCID: https://orcid.org/0000-0002-7270-4328 (2024). Evidence for heterodimerization and functional interaction of the urotensin II and the angiotensin II type 1 receptors Cell Signal , vol. ahead , nº 111056. DOI: 10.1016/j.cellsig.2024.111056. (Sous Presse)

Billard, Étienne; Hébert, Terence E et Chatenet, David ORCID: https://orcid.org/0000-0002-7270-4328 (2023). Exploration of the Urocontrin a Scaffold Yields New Urotensinergic System Allosteric Modulator and Competitive Antagonists Biochemical Pharmacology , vol. 211 , nº 115485. pp. 1-10. DOI: 10.1016/j.bcp.2023.115485.

Nassour, Hassan; Hoang, Tuan Anh; Martin, Ryan D; Dallagnol, Juliana C; Billard, Étienne; Létourneau, Myriam; Novellino, Ettore; Carotenuto, Alfonso; Allen, Bruce G.; Tanny, Jason C; Fournier, Alain; Hébert, Terence E et Chatenet, David ORCID: https://orcid.org/0000-0002-7270-4328 (2021). Lipidated peptides derived from intracellular loops 2 and 3 of the urotensin II receptor act as biased allosteric ligands Journal of Biological Chemistry , vol. 297 , nº 3:101057. pp. 1-19. DOI: 10.1016/j.jbc.2021.101057.

Merlino, Francesco; Billard, Étienne; Yousif, Ali Munaim; Di Maro, Salvatore; Brancaccio, Diego; Abate, Luigi; Carotenuto, Alfonso; Bellavita, Rosa; d'Emmanuele di Villa Bianca, Roberta; Santicioli, Paola; Marinelli, Luciana; Novellino, Ettore; Hébert, Terence E; Lubell, William D; Chatenet, David et Grieco, Paolo (2019). Functional Selectivity Revealed by N-Methylation Scanning of Human Urotensin II and Related Peptides Journal of Medicinal Chemistry , vol. 62 , nº 3. pp. 1455-1467. DOI: 10.1021/acs.jmedchem.8b01601.

Billard, Étienne; Iddir, Mustapha; Nassour, Hassan; Lee-Gosselin, Laura; Poujol de Molliens, Mathilde et Chatenet, David (2019). New directions for urotensin II receptor ligands Peptide Science , vol. 111 , nº e24056. pp. 1-9. DOI: 10.1002/pep2.24056.

Billard, Étienne; Hébert, Terence E et Chatenet, David (2018). Discovery of New Allosteric Modulators of the Urotensinergic System through Substitution of the Urotensin II-Related Peptide (URP) Phenylalanine Residue Journal of Medicinal Chemistry , vol. 61 , nº 19. pp. 8707-8716. DOI: 10.1021/acs.jmedchem.8b00789.

Billard, Étienne; Létourneau, Myriam; Hébert, Terence E et Chatenet, David (2017). Insight into the role of Urotensin II-Related Peptide Tyrosine residue in UT activation Biochemical Pharmacology , vol. 144 . pp. 100-107. DOI: 10.1016/j.bcp.2017.08.003.

Strack, Martin; Billard, Étienne; Chatenet, David et Lubell, William D (2017). Urotensin core mimics that modulate the biological activity of urotensin-II related peptide but not urotensin-II Bioorganic and Medicinal Chemistry Letters , vol. 27 , nº 15. pp. 3412-3416. DOI: 10.1016/j.bmcl.2017.05.088.

Douchez, Antoine; Billard, Étienne; Hébert, Terence E; Chatenet, David et Lubell, William D (2017). Design, Synthesis, and Biological Assessment of Biased Allosteric Modulation of the Urotensin II Receptor Using Achiral 1,3,4-Benzotriazepin-2-one Turn Mimics Journal of Medicinal Chemistry , vol. 60 , nº 23. pp. 9838-9859. DOI: 10.1021/acs.jmedchem.7b01525.

Merlino, Francesco; Yousif, Ali Munaim; Billard, Étienne; Dufour-Gallant, Julien; Turcotte, Stéphane; Grieco, Paolo; Chatenet, David et Lubell, William D (2016). Urotensin II(4-11) Azasulfuryl Peptides: Synthesis and Biological Activity Journal of Medicinal Chemistry , vol. 59 , nº 10. pp. 4740-4752. DOI: 10.1021/acs.jmedchem.6b00108.

Vladoiu, Maria Claudia; Labrie, Marilyne; Létourneau, Myriam; Egesborg, Philippe; Gagné, Donald; Billard, Étienne; Grosset, Andrée-Anne; Doucet, Nicolas ORCID: https://orcid.org/0000-0002-1952-9380; Chatenet, David et St-Pierre, Yves (2015). Design of a peptidic inhibitor that targets the dimer interface of a prototypic galectin Oncotarget , vol. 6 , nº 38. pp. 40970-80. DOI: 10.18632/oncotarget.5403.

Billard, Étienne; Létourneau, Myriam et Chatenet, David . Étude des relations structure-activité sur la position 6 de l’urotensine related peptide. In: 9e édition, Congrès Armand-Frappier 2015, 12-14 novembre 2015, Orford (Québec).

Billard, Étienne; Létourneau, Myriam; Hébert, Terry et Chatenet, David . Mise en lumière du méchanisme d'activation du récepteur UT In: 1ère journée scientifique de l'axe pharmacologie et toxicologie, 28 octobre 2016, INRS- Institut Armand-Frapper, Laval, Qc, Canada.

Billard, Étienne; Létourneau, Myriam; Hébert, Terry et Chatenet, David . Mise en lumière du rôle du résidu Tyr6 de l’Urotensin II-related peptide dans l’activation d’UT In: Congrès Armand-Frappier 2017 (10e édition), 9-11 novembre 2017, Orford (Québec).